Peptide Ligand | Wild Type | Reported Wild Type | L24A | L34A | L24A,L34A |
---|---|---|---|---|---|
[125I-Tyr]CGRP(8–37) | 0.9 ± 0.2 | 0.2a | 9.0 | 9.0 | 9.0 |
CGRP | 1.4 ± 0.3 | 0.4H, 32L a | 8.9 ± 3.1 | 10.8 ± 2.2 | 9.3 ± 2.8 |
AcCGRP(19–37) | 227 ± 86 | 933b | 3000 ± 1400 | 4600 ± 1200 | 2000 ± 1000 |
CGRP(1–36) | > 10,000 | n.d. | > 10,000 | > 10,000 | > 10,000 |
CGRP(1–19) | > 10,000 | n.d. | > 10,000 | > 10,000 | > 10,000 |