Figure 8From: Long-acting κ opioid antagonists nor-BNI, GNTI and JDTic: pharmacokinetics in mice and lipophilicityConcentration-effect relationships derived from Figures 5 and 6. A: Plasma nor-BNI concentrations against reported μ and κ antagonism at the indicated times (mice, 20 mg kg−1 s.c. [10]). B: Plasma and brain JDTic concentrations against reported κ antagonism (mice, i.g. [15]).Back to article page