From: Structural and functional definition of the specificity of a novel caspase-3 inhibitor, Ac-DNLD-CHO
 | Kiapp a (nM) | |||
---|---|---|---|---|
Inhibitor | Caspase-3 | Caspase-7 | Caspase-8 | Caspase-9 |
Ac-DEVD-CHO | 0.288 ± 0.087 | 4.48 ± 0.21 | 0.597 ± 0.095 | 1.35 ± 0.31 |
Ac-DQTD-CHO | 1.27 ± 0.11 | 21.8 ± 1.1 | 9.75 ± 1.09 | 14.5 ± 0.7 |
Ac-DMQD-CHO | 13.3 ± 0.3 | >200 | >200 | >200 |
Ac-DNLD-CHO | 0.680 ± 0.163 | 55.7 ± 6.0 | >200 | >200 |